007 — SL-2026-007

Retatrutide

Triple Receptor Agonist — GIPR / GLP-1R / GCGR

Retatrutide is the most advanced weight-loss peptide in research — activating three receptors simultaneously for fat-loss results that exceed Ozempic and Tirzepatide. Phase 2 trials showed up to 24% body weight reduction in 48 weeks. The next generation is here.

● Low Stock Lyophilized Powder 5 mg / vial COA Included
€94.90
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SKUSL-RETA-5
FormLyophilized Powder
Quantity5 mg / vial
Purity≥98% HPLC
CAS Number2381272‑16‑6
Molecular FormulaC222H376N64O67
Molecular Weight~4800 Da
Storage−20°C, protect from light
Shelf Life24 months (unopened)
ReconstitutionBacteriostatic water or PBS, 1 mg/mL typical
Overview

What is Retatrutide?

Retatrutide is a single synthetic peptide that activates three receptors at once — the GLP-1 receptor (the Ozempic target), the GIP receptor (the Mounjaro addition), and the glucagon receptor. No approved drug does this yet. And the results speak for themselves: Phase 2 trials published in the New England Journal of Medicine showed up to 24% body weight reduction over 48 weeks — substantially more than any approved GLP-1 or dual agonist.

Here's why the triple combination works better. GLP-1R suppresses appetite and stabilizes blood sugar. GIP receptor activation improves insulin sensitivity and modulates fat storage. The glucagon receptor — the novel addition — increases energy expenditure by driving thermogenesis and fat burning. In isolation, glucagon raises blood sugar. But combined with the insulin-promoting effects of GLP-1R and GIPR, that glucose effect is neutralised, while the energy expenditure benefit is preserved. The result: caloric deficit from two directions simultaneously.

Retatrutide is currently in Phase 3 clinical trials. For researchers, it's the most powerful available tool for studying the obesity-related metabolic receptor landscape and the synergistic effects of multi-receptor co-activation. Sharp Labs supplies it as lyophilized powder at ≥98% HPLC purity, with Certificate of Analysis included.

Key Benefits

What it's
known for.

Powerful Weight Loss
Triple receptor activation produces greater fat loss than any single or dual agonist studied to date. Phase 2 trials: up to 24% body weight reduction in 48 weeks — substantially exceeding tirzepatide at equivalent timepoints. Greater reductions in body weight, liver fat, and metabolic biomarkers versus all comparators.
Appetite Suppression
Combines GLP-1R-mediated central satiety signalling with GIPR-driven insulin sensitivity for sustained, powerful appetite reduction throughout the day. The additive satiety effect from two receptor pathways produces greater caloric reduction than either agonist alone.
Metabolic Reset
GCGR activation drives thermogenesis in brown adipose tissue and enhanced fatty acid oxidation in the liver — increasing total energy expenditure at rest. The combination of reduced intake (GLP-1R + GIPR) and increased burn (GCGR) creates a dual-mechanism caloric deficit unique to this compound class.
Blood Sugar Control
Comprehensive glucose management across all three incretin and glucagon pathways: glucose-dependent insulin secretion (GLP-1R), improved peripheral insulin sensitivity (GIPR), and hepatic glucose production modulation (GCGR). Studied in T2D and pre-diabetic models for its potential to address metabolic dysregulation more completely than existing agents.
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